SCHEMBL8613362

SCHEMBL8613362

N=C(NC=O)Nc1cc(-c2ccccc2)nc2cccc(N)c12

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.41
ABCG2 Q9UNQ0 2/20 0.40
ABCB1 P08183 1/20 0.40
ABCC1 P33527 1/20 0.40
ACP1 P24666 3/20 0.39
CYP3A4 P08684 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
GFER P55789 1/20 0.37
ME2 P23368 1/20 0.36
ME1 P48163 1/20 0.36
ME3 Q16798 1/20 0.36
PTGER4 P35408 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PDE10A Q9Y233 1/20 0.36
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617724 0.87 ABCG2 (0.41) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8616263 0.86 ABCB1 (0.40) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8616598 0.86 ABCG2 (0.40) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8618937 0.86 PTGER4 (0.46) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8614064 0.84 ABCB1 (0.50) ABCG2ABCB1ABCC1ACP1MEN1
SCHEMBL8620632 0.84 HPGD (0.44) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8617753 0.83 ACP1 (0.51) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8620896 0.83 MEN1 (0.41) ABCG2ABCB1ABCC1ACP1CYP3A4
SCHEMBL8615866 0.82 ABCB1 (0.39) ABCG2ABCB1ABCC1ACP1MEN1
SCHEMBL8615331 0.82 ALDH1A1 (0.41) ABCG2ABCB1ABCC1ACP1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed