SCHEMBL8614064

SCHEMBL8614064

CC(=O)Nc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.50
ABCC1 P33527 1/20 0.50
ABCG2 Q9UNQ0 1/20 0.50
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
ADORA3 P0DMS8 3/20 0.44
ADORA1 P30542 3/20 0.44
KDM4E B2RXH2 4/20 0.44
PDE10A Q9Y233 1/20 0.44
ALDH1A1 P00352 4/20 0.44
MAPT P10636 2/20 0.44
HPGD P15428 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
RXFP1 Q9HBX9 1/20 0.44
CYP2C19 P33261 1/20 0.44
TP53 P04637 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
STAT1 P42224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619792 0.89 ADORA1 (0.47) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8618123 0.89 ADORA1 (0.47) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8618049 0.87 KDM4E (0.41) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8618937 0.86 PTGER4 (0.46) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8615331 0.85 ALDH1A1 (0.41) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8617724 0.84 ABCG2 (0.41) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8614953 0.84 ALDH1A1 (0.42) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8616263 0.84 ABCB1 (0.40) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8616598 0.84 ABCG2 (0.40) ABCB1ABCC1ABCG2KMT2AMEN1
SCHEMBL8613362 0.84 ACHE (0.41) ABCB1ABCC1ABCG2KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed