SCHEMBL8615331

SCHEMBL8615331

CS(=O)(=O)Nc1cccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
LMNA P02545 2/20 0.41
HSP90AA1 P07900 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ACP1 P24666 2/20 0.40
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
NPC1 O15118 1/20 0.39
JAK2 O60674 1/20 0.39
RAB9A P51151 1/20 0.39
GAA P10253 1/20 0.38
THRB P10828 1/20 0.38
KEAP1 Q14145 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
GFER P55789 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614953 0.90 ALDH1A1 (0.42) ALDH1A1LMNAHSP90AA1KDM4EMAPT
SCHEMBL8613761 0.87 TP53 (0.40) ALDH1A1LMNAHSP90AA1KDM4EMAPT
SCHEMBL8618955 0.87 ACLY (0.41) ACP1ABCB1ABCC1ABCG2MEN1
SCHEMBL8615265 0.86 MRGPRX1 (0.37) ALDH1A1HPGDACP1ABCB1ABCC1
SCHEMBL8617822 0.86 ACLY (0.38) KDM4EMAPTACP1ABCB1ABCC1
SCHEMBL8614064 0.85 ABCB1 (0.50) ALDH1A1KDM4EMAPTHPGDNPSR1
SCHEMBL8619728 0.84 KEAP1 (0.43) ALDH1A1LMNAHSP90AA1KDM4EMAPT
SCHEMBL8618937 0.84 PTGER4 (0.46) ALDH1A1KDM4EACP1ABCB1ABCC1
SCHEMBL8619792 0.83 ADORA1 (0.47) ALDH1A1KDM4EMAPTHPGDACP1
SCHEMBL8618123 0.83 ADORA1 (0.47) ALDH1A1LMNAKDM4EMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed