SCHEMBL8620945

SCHEMBL8620945

COc1ccc2nc(-c3ccccc3)cc(NC(=N)NC=O)c2c1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 5/20 0.56
PLA2G2A P14555 2/20 0.56
KDM4E B2RXH2 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
MEN1 O00255 2/20 0.53
KMT2A Q03164 2/20 0.53
TACR3 P29371 4/20 0.52
NQO1 P15559 1/20 0.49
CA12 O43570 1/20 0.47
CA1 P00915 1/20 0.47
CA2 P00918 1/20 0.47
CA9 Q16790 1/20 0.47
CYP3A4 P08684 1/20 0.47
ABCB1 P08183 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
ALDH1A1 P00352 1/20 0.46
ACP1 P24666 1/20 0.46
ACACA Q13085 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8616497 0.93 TACR3 (0.61) NQO2PLA2G2AKDM4ESMN1; SMN2MEN1
SCHEMBL8620711 0.89 ACP1 (0.60) KDM4EALDH1A1ACP1ACACA
SCHEMBL8615887 0.89 RAB9A (0.47) NQO2PLA2G2AKDM4ESMN1; SMN2MEN1
SCHEMBL8616673 0.88 CA2 (0.50) NQO2PLA2G2AKDM4ESMN1; SMN2MEN1
SCHEMBL8614857 0.87 ABCB1 (0.55) KDM4ESMN1; SMN2MEN1KMT2ATACR3
SCHEMBL8620866 0.87 ALDH1A1 (0.46) NQO2PLA2G2AKDM4ESMN1; SMN2MEN1
SCHEMBL8613853 0.85 ALDH1A1 (0.52) KDM4EMEN1KMT2ACYP3A4ABCB1
SCHEMBL8615676 0.85 ACP1 (0.48) TACR3CYP3A4ABCB1ABCG2ACP1
SCHEMBL8616302 0.84 PDE10A (0.43) NQO2PLA2G2AKDM4ESMN1; SMN2MEN1
SCHEMBL8615684 0.84 ESR1 (0.43) MEN1KMT2ATACR3CYP3A4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed