SCHEMBL8614946

SCHEMBL8614946

CCS(=O)(=O)Nc1cccc2nc(-c3ccccc3)cc(C(=O)NC(=N)N)c12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
MEN1 O00255 6/20 0.43
KMT2A Q03164 6/20 0.43
CYP1A2 P05177 2/20 0.43
ALOX12 P18054 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP3A4 P08684 1/20 0.43
GFER P55789 1/20 0.41
KDM4E B2RXH2 6/20 0.41
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA9 Q16790 2/20 0.41
POLB P06746 1/20 0.41
TACR3 P29371 5/20 0.41
TACR2 P21452 2/20 0.41
CNR1 P21554 2/20 0.41
MAPT P10636 1/20 0.41
PTGER4 P35408 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8615259 0.92 TACR3 (0.42) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8615326 0.90 MEN1 (0.45) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8619780 0.85 ADORA3 (0.47) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8614054 0.84 KMT2A (0.51) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8618942 0.83 ACLY (0.45) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8617819 0.82 ACLY (0.42) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8616347 0.81 ALDH1A1 (0.53) ALDH1A1MEN1KMT2ACYP1A2CYP2C19
SCHEMBL8618116 0.81 ADORA1 (0.47) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8618932 0.81 PTGER4 (0.55) ALDH1A1MEN1KMT2ACYP1A2ALOX12
SCHEMBL8615781 0.81 CA12 (0.44) ALDH1A1MEN1KMT2ACYP1A2ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed