SCHEMBL8615346

SCHEMBL8615346

NCC(N)C(c1ccccc1)C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 4/20 0.46
HTR2A P28223 3/20 0.46
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
DPP4 P27487 2/20 0.39
F2 P00734 1/20 0.39
HRH1 P35367 2/20 0.39
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28745675 0.89 CHRNB2 (0.52) TAAR1HTR2ACHRNB2CHRNA4
SCHEMBL1666957 0.78 GABBR2 (0.47)
SCHEMBL5402204 0.77 DPP4 (0.56) TAAR1HTR2ADPP4F2
SCHEMBL1258400 0.72 TAAR1 (0.52) TAAR1HTR2ACHRNB2CHRNA4DPP4
SCHEMBL6991789 0.72 TAAR1 (0.52) TAAR1HTR2ACHRNB2CHRNA4DPP4
SCHEMBL7291506 0.72 TAAR1 (0.52) TAAR1HTR2ACHRNB2CHRNA4DPP4
SCHEMBL28080494 0.72 TAAR1 (0.52) TAAR1HTR2ACHRNB2CHRNA4DPP4
SCHEMBL4773075 0.72 TAAR1 (0.56) TAAR1HTR2ACHRNB2CHRNA4DPP4
SCHEMBL3640948 0.72 DPP4 (0.62) TAAR1HTR2ACHRNB2CHRNA4DPP4
Iodide SCHEMBL28932197 0.71 TAAR1 (0.50) TAAR1HTR2ACHRNB2CHRNA4HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5786352-A CARDIOVASCULAR DISORDERS, TACHYKININ RECEPTOR ANTAGONIST TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-07-28 US disclosed