SCHEMBL8618277

SCHEMBL8618277

CN1CCC(COc2cc3c(cc2Br)CCN3C(=O)Nc2ccc(-c3ccncc3)c(Cl)c2)CC1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.47
HTR1D P28221 1/20 0.47
HTR1B P28222 1/20 0.47
HTR2C P28335 17/20 0.46
HTR2A P28223 14/20 0.46
HTR2B P41595 8/20 0.45
CYP1A2 P05177 3/20 0.43
SLC2A1 P11166 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8620775 0.93 HTR2C (0.45) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8660110 0.89 CHRNB1 (0.45) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8617192 0.88 HTR1A (0.49) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8618434 0.87 HTR1A (0.46) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8119472 0.81 HTR1A (0.64) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8623325 0.77 HTR2C (0.51) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8137640 0.76 HTR1A (0.63) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8616709 0.75 HTR2C (0.49) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8618094 0.73 HTR1A (0.62) HTR1AHTR1DHTR1BHTR2CHTR2A
SCHEMBL8139246 0.73 HTR1A (0.61) HTR1AHTR1DHTR1BHTR2CHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed