SCHEMBL8620775

SCHEMBL8620775

CN1CCCC(COc2cc3c(cc2Br)CCN3C(=O)Nc2ccc(-c3ccncc3)c(Cl)c2)C1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 16/20 0.45
HTR2A P28223 13/20 0.45
HTR1A P08908 1/20 0.45
HTR1D P28221 1/20 0.45
HTR1B P28222 1/20 0.45
HTR2B P41595 9/20 0.44
CYP1A2 P05177 4/20 0.42
CCR2 P41597 1/20 0.41
KCNH2 Q12809 1/20 0.41
HRH3 Q9Y5N1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618277 0.93 HTR1A (0.47) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8660110 0.89 CHRNB1 (0.45) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8618434 0.88 HTR1A (0.46) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8617192 0.84 HTR1A (0.49) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8119472 0.79 HTR1A (0.64) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8623325 0.75 HTR2C (0.51) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8137640 0.74 HTR1A (0.63) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8616709 0.73 HTR2C (0.49) HTR2CHTR2AHTR1AHTR1DHTR1B
SCHEMBL8621841 0.73 HRH3 (0.44) HRH3
SCHEMBL8139246 0.71 HTR1A (0.61) HTR2CHTR2AHTR1AHTR1DHTR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998050346-A2 ACETAMIDE AND UREA DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THE TREATMENT OF CNS DISORDERS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed