SCHEMBL8618280

SCHEMBL8618280

CC(=O)NCC(C)C(=O)ON1CCC[C@@H](CCc2ccncc2)C1=O

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 1/20 0.34
ITGA2B P08514 1/20 0.34
HRH3 Q9Y5N1 2/20 0.33
FAAH O00519 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP19A1 P11511 1/20 0.33
GFER P55789 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
FKBP1A P62942 1/20 0.32
HTT P42858 1/20 0.32
CHRM3 P20309 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619292 0.85 GPBAR1 (0.34) HSD17B10FKBP1A
SCHEMBL8621103 0.85 ACE (0.34) ITGB3ITGA2BCYP19A1FKBP1ACHRM3
SCHEMBL8617240 0.84 ITGB3 (0.39) ITGB3ITGA2BHSD17B10MEN1KMT2A
SCHEMBL8619325 0.84 MC4R (0.38) ITGB3ITGA2BCYP19A1MEN1KMT2A
SCHEMBL7322436 0.83 HRH3 (0.40) ITGB3ITGA2BHRH3CYP19A1GFER
SCHEMBL8619314 0.82 MTNR1A (0.40) ITGB3ITGA2BCYP19A1MEN1KMT2A
SCHEMBL8621090 0.82 MTNR1A (0.36) ITGB3ITGA2BHSD17B10CYP19A1CHRM3
SCHEMBL8617159 0.82 DPP4 (0.37) ITGB3ITGA2BROCK1
SCHEMBL8619355 0.80 ITGB3 (0.39) ITGB3ITGA2BHRH3FAAHCYP19A1
SCHEMBL8915843 0.78 ITGB3 (0.33) ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852045-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-12-22 US disclosed
US-5773575-A REACTING A CARBOXYLIC ACID AND AMINE WITH COUPLING AGENT MERCK & CO., INC. (US) 1998-06-30 US disclosed
US-5502165-A AMIDATION OF CARBOXY COMPOOUND WITH AMINE IN WATER AND SOLVENT MERCK & CO., INC. (US) 1996-03-26 US disclosed