SCHEMBL8618682

SCHEMBL8618682

COc1ccc(OC)c(-c2cc(NC(=N)NC=O)c3ccccc3n2)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
KDM4E B2RXH2 3/20 0.47
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
POLB P06746 1/20 0.47
ACP1 P24666 4/20 0.47
USP2 O75604 1/20 0.46
HSD17B10 Q99714 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.45
GAA P10253 2/20 0.45
HTT P42858 1/20 0.45
TP53 P04637 2/20 0.44
ALDH1A1 P00352 1/20 0.44
HPGD P15428 1/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
ADORA3 P0DMS8 2/20 0.43
MAPT P10636 1/20 0.43
IGF1R P08069 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618919 0.92 KMT2A (0.58) KDM4EMEN1KMT2APOLBACP1
SCHEMBL8617748 0.90 ACP1 (0.52) KDM4EMEN1KMT2APOLBACP1
SCHEMBL8620711 0.85 ACP1 (0.60) KDM4EACP1HTTALDH1A1HPGD
SCHEMBL8619193 0.84 ADORA3 (0.45) KDM4EMEN1KMT2APOLBACP1
SCHEMBL8614857 0.84 ABCB1 (0.55) KDM4EMEN1KMT2AACP1GAA
SCHEMBL8614845 0.84 DHODH (0.57) KDM4EMEN1KMT2APOLBGAA
SCHEMBL8619356 0.83 ACP1 (0.42) MEN1KMT2APOLBACP1GAA
SCHEMBL8615676 0.83 ACP1 (0.48) ACP1
SCHEMBL8616497 0.82 TACR3 (0.61) KDM4EMEN1KMT2AACP1HTT
SCHEMBL8619346 0.82 TACR3 (0.46) CYP2D6CYP2C9KDM4EGAATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed