SCHEMBL8619356

SCHEMBL8619356

COc1cccc(OC)c1-c1cc(NC(=N)NC=O)c2ccccc2n1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 4/20 0.42
ABCB1 P08183 2/20 0.42
ABCG2 Q9UNQ0 2/20 0.42
IGF1R P08069 3/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
GAA P10253 1/20 0.41
ALDH1A1 P00352 2/20 0.40
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DHODH Q02127 2/20 0.39
ABCC1 P33527 1/20 0.39
TRPV1 Q8NER1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8617748 0.89 ACP1 (0.52) ACP1IGF1RHTTMEN1KMT2A
SCHEMBL8619193 0.88 ADORA3 (0.45) ACP1ABCB1ABCG2IGF1RHTT
SCHEMBL8615877 0.85 PTGER4 (0.41) ACP1ABCB1ABCG2HTTMEN1
SCHEMBL8614845 0.85 DHODH (0.57) HTTMEN1KMT2AGAAALDH1A1
SCHEMBL8618682 0.83 CYP2D6 (0.51) ACP1IGF1RHTTMEN1KMT2A
SCHEMBL8618919 0.83 KMT2A (0.58) ACP1MEN1KMT2AGAAALDH1A1
SCHEMBL8614857 0.83 ABCB1 (0.55) ACP1ABCB1ABCG2MEN1KMT2A
SCHEMBL8620711 0.83 ACP1 (0.60) ACP1HTTALDH1A1MAPTHPGD
SCHEMBL8615676 0.83 ACP1 (0.48) ACP1ABCB1ABCG2
SCHEMBL8618203 0.82 HTT (0.40) ACP1ABCB1ABCG2HTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed