SCHEMBL8618919

SCHEMBL8618919

COc1ccc(-c2cc(NC(=N)NC=O)c3ccccc3n2)c(OC)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.58
KDM4E B2RXH2 4/20 0.58
MEN1 O00255 4/20 0.58
POLB P06746 2/20 0.58
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
TDP1 Q9NUW8 1/20 0.49
ACP1 P24666 4/20 0.47
LMNA P02545 3/20 0.47
HPGD P15428 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ALDH1A1 P00352 2/20 0.46
MAPT P10636 2/20 0.45
GAA P10253 1/20 0.45
HSP90AA1 P07900 1/20 0.45
ADORA3 P0DMS8 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8618682 0.92 CYP2D6 (0.51) KMT2AKDM4EMEN1POLBACP1
SCHEMBL8617748 0.90 ACP1 (0.52) KMT2AKDM4EMEN1POLBACP1
SCHEMBL8620711 0.85 ACP1 (0.60) KDM4EACP1LMNAHPGDALDH1A1
SCHEMBL8619193 0.84 ADORA3 (0.45) KMT2AKDM4EMEN1POLBACP1
SCHEMBL8614857 0.84 ABCB1 (0.55) KMT2AKDM4EMEN1TDP1ACP1
SCHEMBL8615676 0.83 ACP1 (0.48) ACP1
SCHEMBL8619356 0.83 ACP1 (0.42) KMT2AMEN1POLBACP1LMNA
SCHEMBL8616497 0.82 TACR3 (0.61) KMT2AKDM4EMEN1TDP1ACP1
SCHEMBL8619346 0.82 TACR3 (0.46) KDM4ECA12CA1CA2CA9
SCHEMBL8616673 0.82 CA2 (0.50) KMT2AKDM4EMEN1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed