SCHEMBL8619003

SCHEMBL8619003

CC(=O)Nc1cccc2c(C(=O)NC(N)=Nc3ccccc3)ccnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC40A1 Q9NP59 3/20 0.46
ADORA2A P29274 1/20 0.44
KDM4E B2RXH2 6/20 0.41
SMN1; SMN2 Q16637 4/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
RAB9A P51151 4/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 2/20 0.39
SCNN1A P37088 1/20 0.39
GMNN O75496 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
HPGD P15428 1/20 0.39
NFKB1 P19838 1/20 0.39
THPO P40225 1/20 0.39
STAT6 P42226 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8613222 0.96 SLC40A1 (0.48) SLC40A1ADORA2AKDM4ESMN1; SMN2MAPT
SCHEMBL8613894 0.86 SLC40A1 (0.42) SLC40A1ADORA2AKDM4ESMN1; SMN2MAPT
SCHEMBL8620942 0.85 HDAC6 (0.42) SLC40A1ADORA2AKDM4EKMT2AALDH1A1
SCHEMBL8613492 0.84 ADORA2A (0.44) SLC40A1ADORA2AKDM4ESMN1; SMN2MAPT
SCHEMBL8616000 0.83 KDM4E (0.58) SLC40A1ADORA2AKDM4ESMN1; SMN2MAPT
SCHEMBL8616703 0.83 PIK3CA (0.47) SLC40A1ADORA2AKDM4ESMN1; SMN2KMT2A
SCHEMBL8614069 0.83 ADORA2A (0.44) ADORA2AKDM4ESMN1; SMN2MAPTKMT2A
SCHEMBL8619905 0.82 SMN1; SMN2 (0.42) SLC40A1ADORA2AKDM4ESMN1; SMN2MAPT
SCHEMBL8618769 0.82 ALDH1A1 (0.47) SLC40A1ADORA2AKDM4ESMN1; SMN2KMT2A
SCHEMBL8617725 0.82 PDE4A (0.46) ADORA2ASMN1; SMN2RAB9AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed