SCHEMBL8620942

SCHEMBL8620942

CCCCCC(=O)Nc1cccc2c(C(=O)NC(N)=Nc3ccccc3)ccnc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.42
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42
CETP P11597 2/20 0.42
SOAT1 P35610 2/20 0.41
TSHR P16473 3/20 0.41
SLC40A1 Q9NP59 2/20 0.41
EP300 Q09472 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619003 0.85 SLC40A1 (0.46) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8613222 0.81 SLC40A1 (0.48) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8613894 0.79 SLC40A1 (0.42) HDAC3HDAC1HDAC2CETPSLC40A1
SCHEMBL8615876 0.79 RPS6KB1 (0.38) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8617422 0.79 SLC40A1 (0.38) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8613484 0.78 RAB9A (0.43) HDAC6HDAC3HDAC4HDAC1HDAC7
SCHEMBL8613492 0.78 ADORA2A (0.44) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8620689 0.78 MEN1 (0.41) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8615118 0.78 SLC40A1 (0.48) SLC40A1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL8616703 0.77 PIK3CA (0.47) SLC40A1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0726254-B1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS (JP) 1998-05-06 EP disclosed
US-5627193-A MEDICAL DIAGNOSIS, CARDIOVASCULAR DIAORDERS AND PROTECTION OF ORGANS FOR TRANSPLANTATION MITSUI TOATSU CHEMICALS, INC. (JP) 1997-05-06 US disclosed
EP-0726254-A1 Quinoline-4-carbonylguanidine derivates, process for producing the same and pharmaceutical preparations containing the compounds MITSUI TOATSU CHEMICALS, Inc. (JP) 1996-08-14 EP disclosed