SCHEMBL8622121

SCHEMBL8622121

CCOC(=O)C1=C(c2ccccc2)c2ccccc2C1c1ccc2c(c1)OCO2

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
TDP1 Q9NUW8 1/20 0.46
PRKCI P41743 1/20 0.45
PRKCZ Q05513 1/20 0.45
TP53 P04637 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
MEN1 O00255 1/20 0.44
USP2 O75604 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
HSD17B10 Q99714 1/20 0.44
MGAM O43451 1/20 0.44
AMY1A P0DUB6 1/20 0.44
GAA P10253 1/20 0.44
SI P14410 1/20 0.44
MGAM2 Q2M2H8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947116 0.94 ALDH1A1 (0.51) ALDH1A1PRKCIPRKCZTP53TSHR
SCHEMBL9204054 0.87 EDNRB (0.44) ALDH1A1MEN1USP2MAPTHPGD
SCHEMBL8625505 0.86 PRKCI (0.47) ALDH1A1PRKCIPRKCZTP53TSHR
SCHEMBL8623769 0.85 EDNRA (0.49) ALDH1A1TDP1PRKCIPRKCZ
SCHEMBL7533335 0.85 MEN1 (0.47) MEN1KMT2A
SCHEMBL8621789 0.84 ABCB1 (0.46) ALDH1A1TDP1PRKCIPRKCZMGAM
SCHEMBL6958031 0.82 KDM4E (0.53) ALDH1A1TDP1MEN1MAPTKMT2A
SCHEMBL8620561 0.81 PRKCI (0.48) ALDH1A1PRKCIPRKCZTP53HSD17B10
SCHEMBL7534280 0.79 PTGS2 (0.47)
SCHEMBL8620425 0.78 ALDH1A1 (0.54) ALDH1A1TDP1TP53MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817693-A Endothelin receptor antagonists SMITHKLINE BEECHAM CORPORATION 1998-10-06 US disclosed
US-5719182-A TREATING HYPERTENSION, RENAL FAILURE, CEREBROVASCULAR DISEASE SMITHKLINE BEECHAM CORPORATION (US) 1998-02-17 US disclosed