SCHEMBL8623769

SCHEMBL8623769

CCOC(=O)C1=C(c2ccc3c(c2)OCO3)c2ccccc2C1c1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 3/20 0.49
EDNRB P24530 1/20 0.49
ALDH1A1 P00352 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
PRKCI P41743 1/20 0.46
PRKCZ Q05513 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7947116 0.91 ALDH1A1 (0.51) ALDH1A1PRKCIPRKCZ
SCHEMBL8621789 0.91 ABCB1 (0.46) EDNRAEDNRBALDH1A1TDP1PRKCI
SCHEMBL8625505 0.90 PRKCI (0.47) ALDH1A1PRKCIPRKCZ
SCHEMBL8678051 0.90 EDNRA (0.52) EDNRAEDNRBALDH1A1
SCHEMBL7531484 0.88 EDNRA (0.56) EDNRAEDNRB
SCHEMBL8620561 0.87 PRKCI (0.48) EDNRAEDNRBALDH1A1PRKCIPRKCZ
SCHEMBL8622121 0.85 ALDH1A1 (0.51) ALDH1A1TDP1PRKCIPRKCZ
SCHEMBL8620425 0.83 ALDH1A1 (0.54) ALDH1A1TDP1
SCHEMBL8626850 0.79 ALDH1A1 (0.47) ALDH1A1TDP1
SCHEMBL7531670 0.78 FABP7 (0.49) EDNRAEDNRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817693-A Endothelin receptor antagonists SMITHKLINE BEECHAM CORPORATION 1998-10-06 US disclosed
US-5719182-A TREATING HYPERTENSION, RENAL FAILURE, CEREBROVASCULAR DISEASE SMITHKLINE BEECHAM CORPORATION (US) 1998-02-17 US disclosed