SCHEMBL8621789

SCHEMBL8621789

CCOC(=O)C1=C(c2ccc3c(c2)OCO3)c2ccccc2C1c1cccc(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.46
ALDH1A1 P00352 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
PRKCI P41743 1/20 0.45
PRKCZ Q05513 1/20 0.45
EDNRB P24530 1/20 0.43
EDNRA P25101 1/20 0.43
SCD5 Q86SK9 1/20 0.42
CTNNB1 P35222 1/20 0.42
WNT3A P56704 1/20 0.42
BCHE P06276 1/20 0.42
MGAM O43451 1/20 0.42
AMY1A P0DUB6 1/20 0.42
GAA P10253 1/20 0.42
SI P14410 1/20 0.42
MGAM2 Q2M2H8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8623769 0.91 EDNRA (0.49) ALDH1A1TDP1PRKCIPRKCZEDNRB
SCHEMBL7947116 0.90 ALDH1A1 (0.51) ALDH1A1PRKCIPRKCZMGAMAMY1A
SCHEMBL7531670 0.88 FABP7 (0.49) EDNRBEDNRA
SCHEMBL8620561 0.85 PRKCI (0.48) ALDH1A1PRKCIPRKCZEDNRBEDNRA
SCHEMBL8625505 0.84 PRKCI (0.47) ALDH1A1PRKCIPRKCZMGAMAMY1A
SCHEMBL8622121 0.84 ALDH1A1 (0.51) ALDH1A1TDP1PRKCIPRKCZMGAM
SCHEMBL8678051 0.81 EDNRA (0.52) ALDH1A1EDNRBEDNRA
SCHEMBL7531484 0.78 EDNRA (0.56) EDNRBEDNRA
SCHEMBL8621791 0.78 EDNRA (0.46) EDNRBEDNRA
SCHEMBL7534280 0.74 PTGS2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5817693-A Endothelin receptor antagonists SMITHKLINE BEECHAM CORPORATION 1998-10-06 US disclosed
US-5719182-A TREATING HYPERTENSION, RENAL FAILURE, CEREBROVASCULAR DISEASE SMITHKLINE BEECHAM CORPORATION (US) 1998-02-17 US disclosed