SCHEMBL8622690

SCHEMBL8622690

CCOC(=O)C(=C(CC)C(=O)O)N(c1ccc(F)c(F)c1F)C1CC1

nearest known ligand 0.33

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.33
EPHX2 P34913 2/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
P2RX7 Q99572 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
MAPT P10636 2/20 0.30
MEN1 O00255 1/20 0.30
LMNA P02545 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
KCNN4 O15554 1/20 0.30
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9128725 0.82 MAPT (0.32) EPHX2ALDH1A1KDM4ETSHRMAPT
SCHEMBL8624411 0.82 OPRD1 (0.39) OPRM1ALDH1A1KDM4ETSHR
SCHEMBL8625380 0.80 MAPT (0.30) MAPTMEN1LMNACYP1A2CYP2C9
SCHEMBL8624414 0.78 OPRM1 (0.33) OPRM1EPHX2
SCHEMBL8626616 0.77 NPSR1 (0.35) OPRM1EPHX2RAB9AALDH1A1KDM4E
SCHEMBL8622686 0.77 NPSR1 (0.35) OPRM1EPHX2RAB9AALDH1A1KDM4E
SCHEMBL8625558 0.73 KMT2A (0.40) EPHX2ALDH1A1P2RX7MAPTMEN1
SCHEMBL8624624 0.71 P2RX7 (0.36) OPRM1P2RX7SIGMAR1
SCHEMBL8622695 0.70
SCHEMBL6651194 0.68 MAPT (0.39) ALDH1A1KDM4ETSHRP2RX7MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
EP-0684942-A4 1995-12-27 EP disclosed
EP-0684942-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1995-12-06 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed
WO-1994019312-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1994-09-01 WO disclosed