SCHEMBL8624624

SCHEMBL8624624

CCC(C(=O)O)=C(C(=O)O)N(c1ccc(F)c(Cl)c1CC)C1CC1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.36
OPRM1 P35372 4/20 0.33
SIGMAR1 Q99720 1/20 0.31
KCNH2 Q12809 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8624414 0.88 OPRM1 (0.33) OPRM1
SCHEMBL8627781 0.82 P2RX7 (0.32) P2RX7
SCHEMBL8622695 0.73
SCHEMBL8622690 0.71 OPRM1 (0.33) P2RX7OPRM1SIGMAR1
SCHEMBL8621817 0.69 ALDH1A1 (0.30)
SCHEMBL8624411 0.64 OPRD1 (0.39) OPRM1
SCHEMBL10528043 0.64 LMNA (0.43) P2RX7OPRM1
SCHEMBL9847891 0.64 KDM4E (0.34) P2RX7KCNH2HRH3
SCHEMBL9084110 0.62 TSHR (0.42)
SCHEMBL91338 0.61 P2RX7 (0.37) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0684942-B1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORP (US) 1998-06-10 EP disclosed
EP-0684942-A4 1995-12-27 EP disclosed
EP-0684942-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1995-12-06 EP disclosed
US-5430152-A Heating aminoarylester in presence of chlorosulfonic acid, oleum HOECHST CELANESE CORPORATION (US) 1995-07-04 US disclosed
WO-1994019312-A1 METHOD FOR PREPARING QUINOLINE CARBOXYLIC ACIDS AND DERIVATIVES THEREOF HOECHST CELANESE CORPORATION (US) 1994-09-01 WO disclosed