SCHEMBL8622964

SCHEMBL8622964

COc1ccc(S(=O)(=O)Nc2ccccc2NC(=O)c2cccnc2C)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.57
ALDH1A1 P00352 4/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
HTT P42858 2/20 0.57
HPGD P15428 2/20 0.57
TP53 P04637 1/20 0.57
L3MBTL1 Q9Y468 1/20 0.57
GLO1 Q04760 1/20 0.57
SLC40A1 Q9NP59 1/20 0.57
POLB P06746 3/20 0.56
KEAP1 Q14145 1/20 0.55
MEN1 O00255 4/20 0.55
KMT2A Q03164 4/20 0.55
MAPT P10636 3/20 0.55
TDP1 Q9NUW8 2/20 0.55
NPC1 O15118 2/20 0.54
KDM4E B2RXH2 1/20 0.54
MAPK1 P28482 1/20 0.54
RECQL P46063 1/20 0.54
TUBB4A P04350 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8627646 0.89 POLB (0.71) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL8627655 0.86 KEAP1 (0.67) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL8626109 0.85 CCR9 (0.66) SMN1; SMN2HPGDGLO1SLC40A1POLB
SCHEMBL8627716 0.84 TUBB4A (0.59) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL8626192 0.83 KEAP1 (0.56) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL6561670 0.83 LMNA (0.55) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL8623537 0.83 KEAP1 (0.56) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL6563193 0.82 ATM (0.56) LMNAALDH1A1SMN1; SMN2HTTHPGD
SCHEMBL8626468 0.81 SMN1; SMN2 (0.69) LMNAALDH1A1SMN1; SMN2L3MBTL1POLB
SCHEMBL6561650 0.81 KEAP1 (0.53) LMNAALDH1A1SMN1; SMN2HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP claimed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP claimed
EP-0472053-B1 Sulfonamide derivatives EISAI CO LTD (JP) 1998-06-17 EP disclosed
US-5610304-A Pyrimidinyl or pyridinyl sulfonamide substituted compounds EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5610320-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-03-11 US disclosed
US-5434172-A Antitumor EISAI CO., LTD. (JP) 1995-07-18 US disclosed
US-5332751-A Antitumor EISAI CO., LTD. (JP) 1994-07-26 US disclosed
US-5292758-A Sulfonamide derivatives EISAI CO., LTD. (JP) 1994-03-08 US disclosed
US-5250549-A Antitumor agents EISAI CO., LTD. (JP) 1993-10-05 US disclosed
EP-0472053-A2 Sulfonamide derivatives Eisai Co., Ltd. (JP) 1992-02-26 EP disclosed