SCHEMBL8629079

SCHEMBL8629079

Cc1ccc(-c2c(-c3ccccc3S(N)(=O)=O)nn(CC#N)c2C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 7/20 0.36
POLB P06746 3/20 0.35
CYP2C9 P11712 4/20 0.35
CYP2C19 P33261 3/20 0.35
MAPT P10636 1/20 0.35
CA12 O43570 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
HPGD P15428 3/20 0.34
CYP1A2 P05177 2/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
LRRK2 Q5S007 1/20 0.33
CA1 P00915 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8632173 0.91 F10 (0.36) F10POLBCYP2C9CYP2C19MAPT
SCHEMBL8629956 0.90 PTGS2 (0.37) F10POLBCYP2C9CYP2C19MAPT
SCHEMBL8630040 0.89 POLB (0.36) F10POLBCYP2C9CYP2C19CA12
SCHEMBL8635045 0.88 PDE9A (0.42) F10POLBCYP2C9CYP2C19MAPT
SCHEMBL8634745 0.86 PTGS2 (0.38) F10POLBCYP2C9CYP2C19MAPT
SCHEMBL8633375 0.86 F10 (0.37) F10POLBCA2CA9LRRK2
SCHEMBL8633822 0.85 POLB (0.33) F10POLBCYP2C9CYP2C19CA12
SCHEMBL8632205 0.85 PTGS2 (0.45) F10POLBCYP2C9CA12CA2
SCHEMBL7779815 0.83 PTGS2 (0.47) CYP2C9CA12CA2CA9CYP3A4
SCHEMBL8629948 0.82 PTGS2 (0.45) F10ALDH1A1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed