SCHEMBL8633822

SCHEMBL8633822

Cc1ccc(-c2c(-c3ccccc3S(N)(=O)=O)nn(CC#N)c2C(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.33
PTGS1 P23219 1/20 0.33
PTGS2 P35354 1/20 0.33
F10 P00742 6/20 0.33
ALOX5AP P20292 4/20 0.33
FEN1 P39748 4/20 0.33
CA12 O43570 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
ALDH1A1 P00352 1/20 0.32
KDM4E B2RXH2 2/20 0.32
HPGD P15428 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
LRRK2 Q5S007 1/20 0.32
NPSR1 Q6W5P4 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8635408 0.90 PTGS2 (0.36) POLBPTGS1PTGS2F10ALOX5AP
SCHEMBL8629841 0.88 PTGS2 (0.39) PTGS1PTGS2F10ALOX5APFEN1
SCHEMBL8630040 0.87 POLB (0.36) POLBPTGS2F10ALOX5APFEN1
SCHEMBL8628877 0.85 PTGS2 (0.42) POLBPTGS1PTGS2ALDH1A1KDM4E
SCHEMBL8629079 0.85 F10 (0.36) POLBPTGS2F10CA12CA2
SCHEMBL8632205 0.84 PTGS2 (0.45) POLBPTGS1PTGS2F10ALOX5AP
SCHEMBL8630167 0.84 PTGS2 (0.44) PTGS1PTGS2F10ALOX5APFEN1
SCHEMBL7780500 0.84 PTGS2 (0.47) PTGS1PTGS2CA12CA2CA9
SCHEMBL8631787 0.83 PTGS2 (0.40) POLBPTGS2F10CA2CA9
SCHEMBL8633375 0.83 F10 (0.37) POLBPTGS2F10CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed