SCHEMBL8629980

SCHEMBL8629980

CC(C)(C)[Si](C)(C)OCCc1c([Si](C)(C)C)[nH]c2ccc([N+](=O)[O-])cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
PKM P14618 1/20 0.41
NPY1R P25929 1/20 0.41
NPY2R P49146 1/20 0.41
KCNH2 Q12809 1/20 0.40
CTSV O60911 3/20 0.40
CTSL P07711 3/20 0.40
MAPT P10636 4/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA2 P47869 1/20 0.39
LMNA P02545 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL797881 0.94 ALDH1A1 (0.42) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL6595669 0.76 CYP19A1 (0.41) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL5171836 0.74 ALDH1A1 (0.43) ALDH1A1PKMMAPTLMNAKDM4E
SCHEMBL8629985 0.74 CTSV (0.38) ALDH1A1MEN1KMT2APOLBPKM
SCHEMBL4349844 0.73 KIF11 (0.39) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL2367117 0.72 TSHR (0.47) ALDH1A1KMT2APOLBKCNH2MAPT
SCHEMBL4350279 0.71 HCRTR1 (0.48) ALDH1A1MEN1KMT2APOLBMAPT
SCHEMBL23882981 0.71 HSD17B10 (0.43) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL30001627 0.71 HSD17B10 (0.43) ALDH1A1MEN1KMT2AMAPTLMNA
SCHEMBL4350293 0.69 HTR1D (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644187-B1 Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL MYERS SQUIBB CO (US) 1998-07-01 EP disclosed
EP-0644187-A1 Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL-MYERS SQUIBB COMPANY (US) 1995-03-22 EP disclosed
US-5382592-A Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US disclosed