SCHEMBL8629985

SCHEMBL8629985

C[SiH](C)OC(Cc1c([Si](C)(C)C)[nH]c2ccc([N+](=O)[O-])cc12)C(C)(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 4/20 0.38
CTSL P07711 4/20 0.38
CA12 O43570 2/20 0.37
CA9 Q16790 2/20 0.37
MAPT P10636 4/20 0.37
ALDH1A1 P00352 3/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
POLB P06746 1/20 0.37
PKM P14618 1/20 0.37
NPY1R P25929 1/20 0.37
NPY2R P49146 1/20 0.37
GFER P55789 1/20 0.37
GABRA1 P14867 1/20 0.37
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA2 P47869 1/20 0.37
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8629977 0.78 CTSV (0.40) CTSVCTSLCA12CA9MAPT
SCHEMBL8629980 0.74 ALDH1A1 (0.41) CTSVCTSLCA12CA9MAPT
SCHEMBL797881 0.72 ALDH1A1 (0.42) CTSVCTSLCA12CA9MAPT
SCHEMBL7006659 0.64 HTT (0.45) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL7471041 0.63 KMT2A (0.52) MAPTALDH1A1MEN1KMT2APOLB
SCHEMBL8472554 0.63 CHRNB2 (0.49) MAPTALDH1A1MEN1KMT2APOLB
SCHEMBL7472196 0.63 KMT2A (0.44) MAPTALDH1A1MEN1KMT2APOLB
SCHEMBL1780014 0.63 CA12 (0.46) CTSVCTSLCA12CA9MAPT
SCHEMBL29540314 0.63 GABRA1 (0.70) CTSVCTSLCA12CA9MAPT
SCHEMBL155013 0.63 GABRA1 (0.70) CTSVCTSLCA12CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644187-B1 Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL MYERS SQUIBB CO (US) 1998-07-01 EP disclosed
EP-0644187-A1 Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL-MYERS SQUIBB COMPANY (US) 1995-03-22 EP disclosed
US-5382592-A Antimigraine cyclobutenedione derivatives of tryptamines BRISTOL-MYERS SQUIBB COMPANY (US) 1995-01-17 US disclosed