SCHEMBL8630165

SCHEMBL8630165

COc1ccc(-c2c(NS(=O)(=O)c3ccccc3)nn(CC#N)c2C(F)F)cc1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 5/20 0.39
PI4KB Q9UBF8 4/20 0.38
SCN9A Q15858 1/20 0.38
PTGS2 P35354 4/20 0.38
PTGS1 P23219 2/20 0.38
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HTR6 P50406 1/20 0.37
EDNRA P25101 1/20 0.37
KDM1A O60341 1/20 0.37
KCNH2 Q12809 1/20 0.37
PPARA Q07869 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
STAT3 P40763 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631448 0.89 SMN1; SMN2 (0.40) ACLYPI4KBPTGS2PTGS1ABCB11
SCHEMBL8629938 0.89 ACLY (0.41) ACLYPI4KBSCN9APTGS2PTGS1
SCHEMBL8629945 0.88 ACLY (0.43) ACLYPI4KBSCN9APTGS2PTGS1
SCHEMBL8635131 0.88 PI4KB (0.43) ACLYPI4KBPTGS2PTGS1ABCB11
SCHEMBL8627805 0.86 PI4KB (0.38) ACLYPI4KBPTGS2PTGS1ABCB11
SCHEMBL8631946 0.86 ACLY (0.39) ACLYPI4KBSCN9APTGS2PTGS1
SCHEMBL8632809 0.86 PI4KB (0.42) ACLYPI4KBPTGS2PTGS1ABCB11
SCHEMBL8631722 0.86 PPARA (0.41) ACLYPI4KBSCN9APTGS2PTGS1
SCHEMBL8633819 0.84 KDM4E (0.41) ALDH1A1
SCHEMBL8629870 0.83 NPC1 (0.39) ACLYPI4KBSCN9APTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756530-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G. D. SEARLE & CO. (US) 1998-05-26 US disclosed