SCHEMBL21385141

SCHEMBL21385141

CCOC(=O)C(C)C1CCN(c2ccccc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.45
KDM4E B2RXH2 2/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
GPR119 Q8TDV5 1/20 0.45
L3MBTL1 Q9Y468 3/20 0.44
POLB P06746 2/20 0.44
HTT P42858 1/20 0.44
NOTUM Q6P988 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
GAA P10253 2/20 0.44
TSHR P16473 2/20 0.44
GFER P55789 1/20 0.43
KMT2A Q03164 1/20 0.43
SLC6A2 P23975 1/20 0.43
SLC6A4 P31645 1/20 0.43
SLC6A3 Q01959 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21384573 0.85 ALDH1A1 (0.54) MAPTL3MBTL1POLBALDH1A1GAA
SCHEMBL21397342 0.83 NOTUM (0.50) KDM4ECYP2C9CYP2C19GPR119L3MBTL1
SCHEMBL6750641 0.82 OPRM1 (0.54) CYP2C9ALDH1A1
SCHEMBL8546774 0.81 ACHE (0.56) KDM4EL3MBTL1POLBALDH1A1GAA
SCHEMBL5913512 0.79 MAPT (0.67) MAPTKDM4EL3MBTL1POLBHTT
SCHEMBL11167748 0.79 ALDH1A1 (0.55) MAPTKDM4EL3MBTL1HTTNPSR1
SCHEMBL10369008 0.79 SMN1; SMN2 (0.64) CYP2C9CYP2C19L3MBTL1POLBHTT
SCHEMBL14379228 0.78 ALDH1A1 (0.45) MAPTKDM4EL3MBTL1ALDH1A1TSHR
SCHEMBL25409382 0.78 GAA (0.49) MAPTKDM4ECYP2C9CYP2C19ALDH1A1
SCHEMBL21384587 0.77 CHRNB2 (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117185987-A Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-12-08 CN disclosed
CN-111630048-B Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-09-29 CN disclosed
CN-111630048-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-09-04 CN disclosed
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed