SCHEMBL8632757

SCHEMBL8632757

CC1C=C2c3cc(C(=O)O)ccc3C(C)(C)CC21

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.41
RARB P10826 10/20 0.40
RARG P13631 10/20 0.40
RARA P10276 7/20 0.40
CYP26A1 O43174 2/20 0.40
CYP26B1 Q9NR63 1/20 0.40
RXRA P19793 12/20 0.40
RXRB P28702 10/20 0.40
RXRG P48443 7/20 0.40
TDP2 O95551 1/20 0.40
CYP3A4 P08684 1/20 0.37
CRABP2 P29373 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8895391 0.89 MAPT (0.40) AKR1B1RARBRARGCYP26A1CYP26B1
SCHEMBL8563483 0.84 RXRA (0.32) RXRARXRBRXRG
SCHEMBL7118667 0.81 RXRA (0.33) RARBRARGRARACYP26A1CYP26B1
SCHEMBL8892445 0.78 MAPT (0.43) AKR1B1RARBRARGCYP26A1CYP26B1
SCHEMBL8771776 0.76 RARB (0.43) AKR1B1RARBRARGRARACYP26A1
SCHEMBL1071564 0.71 RXRA (0.46) AKR1B1RARBRARGRARACYP26A1
SCHEMBL485022 0.69 TDP2 (0.50) RARBRARGRARACYP26A1CYP26B1
SCHEMBL8771833 0.67 RARB (0.52) RARBRARGRARARXRA
SCHEMBL13189905 0.67 KDM1A (0.46) RARBRARGRARACYP26A1CYP26B1
SCHEMBL6292577 0.67 RARB (0.51) RARBRARGRARACYP26A1CYP26B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773594-A TREATING SKIN DISORDERS, REDUCING SIDE EFFECTS OF OTHER RETINOIDS ALLERGAN (US) 1998-06-30 US disclosed
WO-1997048672-A2 SUBSTITUTED TETRAHYDRONAPHTHALENE AND DIHYDRONAPHTHALENE DERIVATIVES HAVING RETINOID AND/OR RETINOID ANTAGONIST-LIKE BIOLOGICAL ACTIVITY ALLERGAN SALES, INC. (US) 1997-12-24 WO disclosed