SCHEMBL8632877

SCHEMBL8632877

C=COc1ccccc1S(=O)(=O)c1ccccc1C(N)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.44
IRAK4 Q9NWZ3 1/20 0.43
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
CTNNB1 P35222 1/20 0.41
MAPT P10636 2/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA5A P35218 1/20 0.36
CA9 Q16790 1/20 0.36
KMT2A Q03164 2/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 1/20 0.35
NR1I2 O75469 1/20 0.35
LMNA P02545 1/20 0.35
CHRM2 P08172 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28191444 0.81 KDM4E (0.58) KDM4EIRAK4CTNNB1MAPTALDH1A1
SCHEMBL3387938 0.76 CA2 (0.47) CA1CA2CA5ACA9
SCHEMBL30269713 0.76 CA2 (0.47) CA1CA2CA5ACA9
SCHEMBL2723950 0.74 MYC (0.37) MAPTALDH1A1TSHRHSD17B10KMT2A
SCHEMBL8632882 0.73 HTR6 (0.41) KDM4EHTR2AHTR2CCTNNB1ALDH1A1
Potassium Ion SCHEMBL11687702 0.73 ELANE (0.35) HTR6
Bromide SCHEMBL11100956 0.73 MYC (0.36) MAPTALDH1A1TSHRHSD17B10KMT2A
SCHEMBL28440193 0.73 MYC (0.36) MAPTALDH1A1TSHRHSD17B10KMT2A
SCHEMBL8997308 0.72 BCAT2 (0.62) KDM4EHTR2AHTR2CMAPTALDH1A1
SCHEMBL3641319 0.71 ALDH1A1 (0.45) KDM4EHTR2AHTR2CMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0748312-B1 BICYCLIC CARBAMATES AS LEUKOTRIENE D4 ANTAGONISTS PFIZER (US) 1998-07-22 EP claimed
EP-0748312-B1 BICYCLIC CARBAMATES AS LEUKOTRIENE D4 ANTAGONISTS PFIZER (US) 1998-07-22 EP disclosed