SCHEMBL8634397

SCHEMBL8634397

COC(=O)[C@@H]1CCCN1C(=O)C(=O)C1CCCN(C(=O)c2ccc([N+](=O)[O-])cc2Cl)c2ccc(F)cc21

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
WDR5 P61964 1/20 0.41
MAPT P10636 7/20 0.39
ALDH1A1 P00352 6/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
AVPR2 P30518 1/20 0.35
AVPR1A P37288 1/20 0.35
NPC1 O15118 1/20 0.34
LMNA P02545 2/20 0.34
MAPK1 P28482 1/20 0.34
KCNK3 O14649 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
ALOX5 P09917 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633381 0.88 ALDH1A1 (0.39) ALDH1A1AVPR2AVPR1AKCNK3MEN1
SCHEMBL4682740 0.85 ALDH1A1 (0.43) WDR5MAPTALDH1A1SMN1; SMN2AVPR2
SCHEMBL7344728 0.77 ALDH1A1 (0.40) WDR5MAPTALDH1A1SMN1; SMN2LMNA
SCHEMBL7336618 0.74 PKM (0.42) WDR5MAPTALDH1A1SMN1; SMN2AVPR2
SCHEMBL4697134 0.73 ALDH1A1 (0.46) ALDH1A1AVPR2AVPR1AKCNK3GAA
SCHEMBL4684984 0.72 AVPR2 (0.49) WDR5MAPTALDH1A1SMN1; SMN2AVPR2
SCHEMBL4686745 0.71 ALDH1A1 (0.41) WDR5MAPTALDH1A1SMN1; SMN2AVPR2
SCHEMBL4684773 0.71 AVPR2 (0.46) WDR5MAPTALDH1A1SMN1; SMN2AVPR2
SCHEMBL8634401 0.70 MAPT (0.36) WDR5MAPTALDH1A1SMN1; SMN2NPC1
SCHEMBL7333794 0.70 ALDH1A1 (0.41) WDR5MAPTALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed