SCHEMBL7344728

SCHEMBL7344728

O=C(O)[C@@H]1CCCN1C(=O)COC1CCCN(C(=O)c2ccc([N+](=O)[O-])cc2Cl)c2ccc(F)cc21

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
WDR5 P61964 1/20 0.38
CPT2 P23786 1/20 0.37
CPT1A P50416 1/20 0.37
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.35
SLC6A9 P48067 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4682740 0.92 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2WDR5CPT2CPT1A
SCHEMBL7336774 0.88 SLC6A9 (0.36) ALDH1A1SLC6A9
SCHEMBL7336618 0.81 PKM (0.42) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
SCHEMBL4697134 0.79 ALDH1A1 (0.46) ALDH1A1
SCHEMBL8634397 0.77 WDR5 (0.41) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
SCHEMBL7342308 0.76 MAPT (0.39) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
SCHEMBL4681210 0.75 MAPT (0.38) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
SCHEMBL4684092 0.74 WDR5 (0.36) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
Iodide SCHEMBL4686142 0.72 AVPR2 (0.40) ALDH1A1SMN1; SMN2WDR5MAPTLMNA
SCHEMBL5474822 0.72 MAPT (0.39) ALDH1A1SMN1; SMN2WDR5MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514667-B1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMA CO LTD (JP) 1995-08-09 EP disclosed
EP-0514667-A1 Benzazepin derivatives as vasopressin antagonists OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-25 EP disclosed