SCHEMBL8634401

SCHEMBL8634401

COC(=O)[C@@H]1CCCN1C(=O)C(OC1CCCNc2ccc(F)cc21)C(=O)c1ccc([N+](=O)[O-])cc1Cl

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.36
NPC1 O15118 1/20 0.35
WDR5 P61964 1/20 0.35
ALDH1A1 P00352 4/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
KCNK3 O14649 1/20 0.32
GAA P10253 2/20 0.31
ALOX5 P09917 1/20 0.31
P2RX7 Q99572 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
FPR2 P25090 1/20 0.31
SCN9A Q15858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8631703 0.89 KCNK3 (0.33) ALDH1A1KCNK3GAAALOX5P2RX7
SCHEMBL4682740 0.73 ALDH1A1 (0.43) MAPTWDR5ALDH1A1SMN1; SMN2P2RX7
SCHEMBL8634397 0.70 WDR5 (0.41) MAPTNPC1WDR5ALDH1A1SMN1; SMN2
SCHEMBL7344728 0.65 ALDH1A1 (0.40) MAPTWDR5ALDH1A1SMN1; SMN2
SCHEMBL7336618 0.64 PKM (0.42) MAPTNPC1WDR5ALDH1A1SMN1; SMN2
SCHEMBL9727483 0.63 GAA (0.45) ALDH1A1KCNK3GAANPSR1FPR2
SCHEMBL14256154 0.61 HCRTR2 (0.35)
SCHEMBL15962162 0.61 MAPT (0.52) MAPTNPC1ALDH1A1SMN1; SMN2HTT
SCHEMBL6173457 0.61 MAPT (0.52) MAPTNPC1ALDH1A1SMN1; SMN2HTT
SCHEMBL4697134 0.61 ALDH1A1 (0.46) ALDH1A1KCNK3GAAP2RX7SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753644-A Vasopressin antagonist and oxytocin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1998-05-19 US disclosed