SCHEMBL4697134

SCHEMBL4697134

COC(=O)[C@@H]1CCCN1C(=O)COC1CCCN(C(=O)c2ccc(N)cc2Cl)c2ccc(F)cc21

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
AVPR2 P30518 7/20 0.36
P2RX7 Q99572 1/20 0.36
AVPR1A P37288 3/20 0.36
KCNK3 O14649 1/20 0.35
JAK3 P52333 1/20 0.35
BTK Q06187 1/20 0.35
CNR2 P34972 2/20 0.34
GAA P10253 1/20 0.34
CNR1 P21554 1/20 0.34
LOX P28300 1/20 0.34
OXTR P30559 1/20 0.34
PDK2 Q15119 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7336774 0.91 SLC6A9 (0.36) ALDH1A1AVPR2P2RX7AVPR1AOXTR
SCHEMBL4682740 0.88 ALDH1A1 (0.43) ALDH1A1AVPR2P2RX7AVPR1A
SCHEMBL8633381 0.84 ALDH1A1 (0.39) ALDH1A1AVPR2P2RX7AVPR1AKCNK3
SCHEMBL7343891 0.81 AVPR2 (0.42) ALDH1A1AVPR2P2RX7AVPR1AOXTR
SCHEMBL7344728 0.79 ALDH1A1 (0.40) ALDH1A1
SCHEMBL8634397 0.73 WDR5 (0.41) ALDH1A1AVPR2AVPR1AKCNK3GAA
SCHEMBL8631703 0.72 KCNK3 (0.33) ALDH1A1P2RX7KCNK3GAASCN9A
SCHEMBL4685307 0.71 AVPR2 (0.45) ALDH1A1AVPR2
SCHEMBL7336618 0.71 PKM (0.42) ALDH1A1AVPR2AVPR1A
SCHEMBL4688323 0.71 AVPR2 (0.44) ALDH1A1AVPR2AVPR1ASCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902717-A2 Vasopressin antagonist and oxytocin antagonist Otsuka Pharmaceutical Company, Limited (JP) 2008-03-26 EP disclosed
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed
EP-0620003-A1 VASOPRESSIN ANTAGONIST AND OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-10-19 EP disclosed
US-5244898-A Vasopressin antagonist OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-09-14 US disclosed