SCHEMBL8686282

SCHEMBL8686282

CCC(C)S(=O)(=O)NC1CN(c2ccncc2)CCN1C(CCC(=O)OC)Oc1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.35
ITGB3 P05106 2/20 0.34
ITGA2B P08514 2/20 0.34
TSHR P16473 2/20 0.33
HSD17B10 Q99714 1/20 0.33
KCNA5 P22460 2/20 0.32
F10 P00742 4/20 0.32
SMN1; SMN2 Q16637 3/20 0.31
CYP2C9 P11712 2/20 0.31
ALDH1A1 P00352 2/20 0.31
CYP2D6 P10635 1/20 0.31
MAPK1 P28482 1/20 0.31
HIF1A Q16665 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
ACACB O00763 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
CA12 O43570 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8630686 0.94 ITGB3 (0.37) ROCK2ITGB3ITGA2BTSHRHSD17B10
SCHEMBL8697195 0.81 ROCK2 (0.38) ROCK2ITGB3ITGA2BTSHRHSD17B10
SCHEMBL8633129 0.80 KDM4D (0.35) ROCK2ITGB3ITGA2BTSHRF10
SCHEMBL8698839 0.75 FAAH (0.37) ITGB3ITGA2BTSHRHSD17B10F10
SCHEMBL7450096 0.73 ITGB3 (0.42) ROCK2ITGB3ITGA2BTSHRHSD17B10
SCHEMBL8635810 0.73 NPSR1 (0.34) ITGB3ITGA2BTSHRHSD17B10F10
SCHEMBL7398021 0.72 ITGB3 (0.39) ROCK2ITGB3ITGA2BTSHRHSD17B10
SCHEMBL8699716 0.72 F10 (0.36) ITGB3ITGA2BTSHRHSD17B10F10
SCHEMBL27442362 0.70 GAA (0.43) ROCK2ITGB3ITGA2BTSHRHSD17B10
SCHEMBL7403452 0.69 ITGB3 (0.37) ITGB3ITGA2BTSHRF10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed