SCHEMBL8633129

SCHEMBL8633129

COC(=O)CCC(Oc1ccccc1)N1CCN(c2ccncc2)CC1NC(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4D Q6B0I6 3/20 0.35
ROCK2 O75116 1/20 0.34
CKS1B P61024 1/20 0.33
SKP1 P63208 1/20 0.33
SKP2 Q13309 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
NR1H2 P55055 3/20 0.33
NR1H3 Q13133 3/20 0.33
KMT2A Q03164 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ALDH1A1 P00352 1/20 0.32
GAA P10253 1/20 0.32
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
BUB1 O43683 1/20 0.32
DRD2 P14416 3/20 0.32
F10 P00742 1/20 0.32
DRD3 P35462 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8697195 0.82 ROCK2 (0.38) ROCK2ITGB3ITGA2BALDH1A1GAA
SCHEMBL8686282 0.80 ROCK2 (0.35) ROCK2ITGB3ITGA2BALDH1A1TSHR
SCHEMBL7450096 0.74 ITGB3 (0.42) ROCK2ITGB3ITGA2BALDH1A1TSHR
SCHEMBL8698839 0.74 FAAH (0.37) ITGB3ITGA2BALDH1A1GAATSHR
SCHEMBL8630686 0.73 ITGB3 (0.37) ROCK2ITGB3ITGA2BALDH1A1TSHR
SCHEMBL7398021 0.72 ITGB3 (0.39) ROCK2ITGB3ITGA2BALDH1A1TSHR
SCHEMBL8699716 0.71 F10 (0.36) ITGB3ITGA2BALDH1A1GAATSHR
SCHEMBL8635810 0.71 NPSR1 (0.34) ITGB3ITGA2BKMT2AALDH1A1GAA
SCHEMBL7403452 0.70 ITGB3 (0.37) ITGB3ITGA2BALDH1A1TSHRF10
SCHEMBL8634865 0.69 GAA (0.38) ROCK2KMT2AL3MBTL1GAATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed