SCHEMBL8634908

SCHEMBL8634908

N=C(N)NC(=O)c1ccccc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.50
NPC1 O15118 4/20 0.50
ALDH1A1 P00352 8/20 0.48
HSD17B10 Q99714 2/20 0.48
CFTR P13569 1/20 0.48
KDM4E B2RXH2 8/20 0.47
FADS1 O60427 2/20 0.47
GAA P10253 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MAPT P10636 2/20 0.46
HPGD P15428 3/20 0.45
PTGS1 P23219 1/20 0.45
P2RX1 P51575 1/20 0.44
CASP3 P42574 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
PIK3CA P42336 1/20 0.44
POLB P06746 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3070336 0.88 ALDH1A1 (0.42) NPC1ALDH1A1HSD17B10KDM4EGAA
SCHEMBL5574637 0.84 FADS1 (0.54) RAB9ANPC1ALDH1A1HSD17B10CFTR
SCHEMBL28193055 0.81 ALDH1A1 (0.48) RAB9ANPC1ALDH1A1HSD17B10CFTR
SCHEMBL23875051 0.81 CA1 (0.58) RAB9ANPC1ALDH1A1HSD17B10KDM4E
SCHEMBL1242360 0.79 MEN1 (0.53) RAB9ANPC1ALDH1A1HSD17B10KDM4E
SCHEMBL6651792 0.79 HPGD (0.53) RAB9ANPC1ALDH1A1KDM4ESMN1; SMN2
SCHEMBL8416208 0.79 POLB (0.60) RAB9ANPC1ALDH1A1KDM4EGAA
SCHEMBL27393236 0.79 NPC1 (0.62) RAB9ANPC1ALDH1A1KDM4EGAA
SCHEMBL3073042 0.78 PLAU (0.39) NPC1ALDH1A1HSD17B10KDM4EGAA
SCHEMBL6999516 0.78 ALDH1A1 (0.55) RAB9ANPC1ALDH1A1HSD17B10CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1058001-C 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 2000-11-01 CN claimed
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US claimed
US-5696167-A 4-mercaptobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-12-09 US claimed
CN-1134413-A 4-Mercaptobenzoylguanidine derivatives MERCK PATENT GMBH (DE) 1996-10-30 CN claimed
EP-0603650-B1 3,5-Substituted amino benzoylguanidines, process for their preparation, their use as medicine or diagnostic agent, as well as a medicine containing them HOECHST AG (DE) 1997-04-02 EP disclosed
US-5516805-A 3,5-substituted aminobenzoylguanidines, their use as a medicament or diagnostic and medicament containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-05-14 US disclosed
EP-0603650-A1 3,5-Substituted amino benzoylguanidines, process for their preparation, their use as medicine or diagnostic agent, as well as a medicine containing them HOECHST AKTIENGESELLSCHAFT (DE) 1994-06-29 EP disclosed