SCHEMBL6999516

SCHEMBL6999516

CC(=O)NC(=O)c1ccccc1N

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 10/20 0.55
HSD17B10 Q99714 5/20 0.55
CFTR P13569 1/20 0.55
KDM4E B2RXH2 10/20 0.53
HPGD P15428 6/20 0.50
RAB9A P51151 3/20 0.50
POLB P06746 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPC1 O15118 2/20 0.49
CASP3 P42574 1/20 0.49
SENP8 Q96LD8 1/20 0.49
SENP7 Q9BQF6 1/20 0.49
SENP6 Q9GZR1 1/20 0.49
FADS1 O60427 2/20 0.49
GLA P06280 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47
RCE1 Q9Y256 1/20 0.46
PTGS1 P23219 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6366964 0.82 ALDH1A1 (0.53) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL5574637 0.82 FADS1 (0.54) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL8477209 0.80 SIRT2 (0.47) ALDH1A1HSD17B10KDM4EHPGDPOLB
SCHEMBL375579 0.79 ALDH1A1 (0.59) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL9921278 0.79 KDM4E (0.60) ALDH1A1HSD17B10CFTRKDM4EHPGD
Acetic Acid SCHEMBL28650473 0.78 KDM4E (0.56) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL8634908 0.78 RAB9A (0.50) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL5807531 0.78 MAPT (0.60) ALDH1A1HSD17B10CFTRKDM4ERAB9A
SCHEMBL28193055 0.78 ALDH1A1 (0.48) ALDH1A1HSD17B10CFTRKDM4EHPGD
SCHEMBL15361168 0.78 SMN1; SMN2 (0.68) ALDH1A1HSD17B10KDM4EHPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1294707-A2 THIOPHENE DERIVATIVES ACTIVE AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM Pharmacia Italia S.p.A. (IT) 2003-03-26 EP claimed
WO-2001098290-A2 THIOPHENE DERIVATIVES ACTIVE AS KINASE INHIBITORS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM PHARMACIA ITALIA S.P.A. (IT) 2001-12-27 WO claimed
US-6414013-B1 KINASE INHIBITORS; ANTICANCER AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2002-07-02 US disclosed