SCHEMBL8633523

SCHEMBL8633523

CC(=O)C(Oc1ccccc1)(C(=O)O)N1CCN(c2ccnc(C)c2)CC1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.38
PSEN1 P49768 1/20 0.38
PSEN2 P49810 1/20 0.38
APH1B Q8WW43 1/20 0.38
NCSTN Q92542 1/20 0.38
APH1A Q96BI3 1/20 0.38
PSENEN Q9NZ42 1/20 0.38
CHRM1 P11229 1/20 0.37
KMT2A Q03164 1/20 0.36
F10 P00742 2/20 0.35
MAPK1 P28482 2/20 0.35
NPC1 O15118 1/20 0.35
MAPT P10636 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LDHA P00338 1/20 0.34
PPARG P37231 1/20 0.34
CCKAR P32238 1/20 0.34
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8633634 0.85 CYP2C9 (0.46) MAPK1MAPTALDH1A1
SCHEMBL8631971 0.80 ITGB3 (0.40) AOC3KMT2AF10MAPK1MAPT
SCHEMBL8699395 0.78 ALDH1A1 (0.39) KMT2AMAPK1MAPTALDH1A1
SCHEMBL8653961 0.77 PDGFRB (0.52) KMT2AMAPT
SCHEMBL8635770 0.77 ROCK2 (0.49) KMT2AF10MAPK1NPC1MAPT
SCHEMBL8633383 0.77 GPR119 (0.43) CHRM1KMT2AMAPK1NPC1ALDH1A1
SCHEMBL8649587 0.77 NCF1 (0.60) KMT2AMAPK1MAPT
SCHEMBL8635264 0.76 CYP2C9 (0.44) AOC3MAPK1MAPTALDH1A1
SCHEMBL8654165 0.75 PDGFRB (0.33) KMT2AMAPK1NPC1MAPTALDH1A1
SCHEMBL8634909 0.75 KDM4E (0.39) CHRM1MAPK1NPC1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753659-A ANTICOAGULANTS FOR BLOOD DISORDER, CARDIOVASCULAR DISORDER, THROMBOSIS, ZENECA LIMITED (GB) 1998-05-19 US disclosed
US-5750754-A TERTIARY BUTYL 3-METHYL-4-SUBSTITUTED BUTYRATE; CHEMICAL INTERMEDIATES FOR ANTICAOGULANT DRUGS ZENECA LIMITED (GB) 1998-05-12 US disclosed
US-5728701-A INHIBIT PLATELET AGGREGATION ZENECA LIMITED (GB) 1998-03-17 US disclosed