SCHEMBL8635178

SCHEMBL8635178

CCc1cc(Nc2cccc(OC)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.48
AKR1C2 P52895 3/20 0.48
MTNR1B P49286 5/20 0.45
MTNR1A P48039 3/20 0.45
PDE4B Q07343 2/20 0.43
PTGS1 P23219 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
GFER P55789 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
LMNA P02545 1/20 0.43
HPGD P15428 1/20 0.43
NPC1 O15118 2/20 0.42
GAA P10253 2/20 0.42
MAPT P10636 1/20 0.42
RAB9A P51151 1/20 0.42
P2RY2 P41231 2/20 0.41
P2RY4 P51582 2/20 0.41
P2RY12 Q9H244 2/20 0.41
PDE4A P27815 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634230 0.88 AKR1C3 (0.45) AKR1C3AKR1C2PTGS1MEN1KMT2A
SCHEMBL8637536 0.87 AKR1C3 (0.51) AKR1C3AKR1C2MTNR1BMTNR1APDE4B
SCHEMBL8633209 0.85 MEN1 (0.43) AKR1C3AKR1C2PDE4BPTGS1MEN1
SCHEMBL8635140 0.85 BCAT2 (0.42) AKR1C3AKR1C2MEN1KMT2AGFER
SCHEMBL7768696 0.85 PDE4B (0.44) AKR1C3AKR1C2PDE4B
SCHEMBL8632359 0.84 MEN1 (0.44) PTGS1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL8636186 0.82 AKR1C3 (0.44) AKR1C3AKR1C2PTGS1MEN1KMT2A
SCHEMBL8632259 0.82 YAP1 (0.49) AKR1C3AKR1C2LMNAHPGDGAA
SCHEMBL8632351 0.82 PDE4B (0.41) PDE4BPTGS1MEN1KMT2ALMNA
SCHEMBL8635300 0.81 HTT (0.38) PTGS1MAPTP2RY4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed