SCHEMBL8637536

SCHEMBL8637536

COc1cccc(Nc2cc(C)c(C(=O)Cl)cc2S(C)(=O)=O)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 4/20 0.51
AKR1C2 P52895 4/20 0.51
GFER P55789 2/20 0.46
NPC1 O15118 2/20 0.46
GAA P10253 1/20 0.46
PTGS1 P23219 1/20 0.45
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
MEN1 O00255 1/20 0.45
LMNA P02545 1/20 0.45
KMT2A Q03164 1/20 0.45
PDE4B Q07343 1/20 0.45
MTNR1B P49286 2/20 0.44
MTNR1A P48039 1/20 0.43
MAPT P10636 3/20 0.43
RAPGEF4 Q8WZA2 1/20 0.43
PKM P14618 1/20 0.43
HTT P42858 1/20 0.43
IDH1 O75874 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8634936 0.87 AKR1C3 (0.48) AKR1C3AKR1C2SMN1; SMN2MEN1LMNA
SCHEMBL8635178 0.87 AKR1C3 (0.48) AKR1C3AKR1C2GFERNPC1GAA
SCHEMBL8635252 0.85 AKR1C3 (0.50) AKR1C3AKR1C2GFERNPC1PTGS1
SCHEMBL8635463 0.84 AKR1C3 (0.45) AKR1C3AKR1C2GFERGAAMEN1
SCHEMBL7761235 0.84 SLC9A1 (0.55)
SCHEMBL8632908 0.84 PTGS1 (0.43) GAAPTGS1SMN1; SMN2MEN1LMNA
SCHEMBL8635174 0.81 AKR1C3 (0.49) AKR1C3AKR1C2GAAPTGS1SMN1; SMN2
SCHEMBL8632107 0.81 AKR1C3 (0.52) AKR1C3AKR1C2RAPGEF4IDH1
SCHEMBL8634318 0.81 PDE4B (0.46) PTGS1MEN1KMT2APDE4BMAPT
SCHEMBL8633408 0.80 ALDH1A1 (0.39) NPC1PTGS1SMN1; SMN2IDH1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed