SCHEMBL8632259

SCHEMBL8632259

CCc1cc(Nc2cccc(C(F)(F)F)c2)c(S(C)(=O)=O)cc1C(=O)Cl

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
YAP1 P46937 1/20 0.49
TEAD4 Q15561 1/20 0.49
TEAD2 Q15562 1/20 0.49
MPO P05164 4/20 0.47
RXFP1 Q9HBX9 3/20 0.46
IDH1 O75874 1/20 0.46
AKR1C3 P42330 2/20 0.45
AKR1C2 P52895 2/20 0.45
CYP3A4 P08684 4/20 0.43
CYP2C19 P33261 4/20 0.43
CYP2C9 P11712 3/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
IDH2 P48735 1/20 0.43
LMNA P02545 1/20 0.42
GAA P10253 1/20 0.42
CYP2D6 P10635 1/20 0.42
DDR1 Q08345 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7764117 0.88 AKR1C3 (0.42) IDH1AKR1C3AKR1C2CYP3A4CYP2C19
SCHEMBL8632107 0.87 AKR1C3 (0.52) YAP1TEAD4TEAD2MPORXFP1
SCHEMBL8632359 0.86 MEN1 (0.44) LMNAGAA
SCHEMBL7764083 0.85 YAP1 (0.43) YAP1TEAD4TEAD2
SCHEMBL8633209 0.84 MEN1 (0.43) AKR1C3AKR1C2ALDH1A1HPGDLMNA
SCHEMBL8635140 0.84 BCAT2 (0.42) RXFP1AKR1C3AKR1C2CYP3A4CYP2C19
SCHEMBL8635178 0.82 AKR1C3 (0.48) AKR1C3AKR1C2HPGDLMNAGAA
SCHEMBL8632351 0.81 PDE4B (0.41) RXFP1ALDH1A1LMNA
SCHEMBL8633397 0.81 AKR1C3 (0.43) AKR1C3AKR1C2CYP3A4CYP2C19CYP2C9
SCHEMBL8635300 0.80 HTT (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739142-A 4-aminobenzoylguanidine derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-04-14 US disclosed