SCHEMBL8420779

SCHEMBL8420779

CSc1ccc(-c2cc(-c3ccc(SC)cc3)n(NS(=O)(=O)c3ccccc3)n2)cc1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.41
GAA P10253 2/20 0.41
HPGD P15428 1/20 0.41
CYP2C9 P11712 1/20 0.39
MMP2 P08253 2/20 0.39
NPY5R Q15761 1/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP13 P45452 1/20 0.39
MAPT P10636 2/20 0.39
PTGS2 P35354 2/20 0.38
PTGS1 P23219 1/20 0.38
MMP9 P14780 1/20 0.38
TSHR P16473 2/20 0.37
KMT2A Q03164 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
POLB P06746 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A3 P47895 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8420178 0.94 ALDH1A1 (0.42) ALDH1A1GAAHPGDMAPTPTGS2
SCHEMBL8421979 0.94 ALDH1A1 (0.42) ALDH1A1GAAHPGDMAPTPTGS2
SCHEMBL8422371 0.87 MAPT (0.45) ALDH1A1CYP2C9MMP2NPY5RMMP1
SCHEMBL8420749 0.86 MAPT (0.52) ALDH1A1HPGDCYP2C9NPY5RMAPT
SCHEMBL8420791 0.85 GAA (0.43) ALDH1A1GAAHPGDMAPTPTGS2
SCHEMBL8420831 0.85 GAA (0.43) ALDH1A1GAAHPGDPTGS2SMN1; SMN2
SCHEMBL8641068 0.85 PTGS2 (0.53) ALDH1A1GAAHPGDCYP2C9PTGS2
SCHEMBL8636817 0.84 PTGS2 (0.42) ALDH1A1GAAHPGDMMP2MMP1
SCHEMBL8689203 0.84 MMP2 (0.39) ALDH1A1GAAHPGDMMP2MMP1
SCHEMBL8422134 0.84 MAPT (0.51) ALDH1A1GAACYP2C9MMP2NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5908852-A 1,3,5 trisubstituted pyrazole compounds for treatment of inflammation G. D. SEARLE & CO. (US) 1999-06-01 US disclosed