SCHEMBL8637801

SCHEMBL8637801

COc1ccccc1CC1CCN(CCOc2ccccc2)C1

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 2/20 0.56
SIGMAR1 Q99720 2/20 0.56
LTA4H P09960 2/20 0.51
HTR1A P08908 1/20 0.49
SLC6A4 P31645 1/20 0.49
KCNH2 Q12809 2/20 0.48
AURKA O14965 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8640943 0.83 TMEM97 (0.59) TMEM97SIGMAR1LTA4HHTR1ASLC6A4
SCHEMBL8641102 0.80 HTR1A (0.67) TMEM97SIGMAR1LTA4HHTR1ASLC6A4
SCHEMBL1333847 0.79 KCNH2 (0.67) SIGMAR1KCNH2
SCHEMBL8644124 0.78 TMEM97 (0.70) TMEM97SIGMAR1LTA4HHTR1ASLC6A4
Hydrochloric Acid SCHEMBL1332072 0.78 KCNH2 (0.69) SIGMAR1KCNH2
SCHEMBL7032506 0.77 SIGMAR1 (0.75) SIGMAR1KCNH2
SCHEMBL21780869 0.77 TMEM97 (0.63) TMEM97SIGMAR1LTA4HHTR1AKCNH2
Hydrochloric Acid SCHEMBL1333883 0.76 KCNH2 (0.76) SIGMAR1KCNH2
SCHEMBL8639262 0.76 SIGMAR1 (0.70) TMEM97SIGMAR1LTA4HHTR1ASLC6A4
SCHEMBL7375479 0.75 TMEM97 (0.55) TMEM97SIGMAR1LTA4HHTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5723492-A LTA4 hydrolase inhibitor pharmaceutical compositions and methods of use G.D. SEARLE & CO. (US) 1998-03-03 US disclosed
US-5719306-A ANTIINFLAMMATORY AGENTS G.D. SEARLE & CO. (US) 1998-02-17 US disclosed