SCHEMBL8645683

SCHEMBL8645683

COC(=O)C1(C(=O)O)Cc2cc(Br)ccc2N1C(C)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 4/20 0.37
NOTUM Q6P988 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
TUBB4A P04350 1/20 0.36
TUBB P07437 1/20 0.36
TUBA3C P0DPH7 1/20 0.36
TUBA1B P68363 1/20 0.36
TUBA4A P68366 1/20 0.36
TUBB4B P68371 1/20 0.36
TUBB3 Q13509 1/20 0.36
TUBB2A Q13885 1/20 0.36
TUBB8 Q3ZCM7 1/20 0.36
TUBA3E Q6PEY2 1/20 0.36
TUBA1A Q71U36 1/20 0.36
TUBA1C Q9BQE3 1/20 0.36
TUBB6 Q9BUF5 1/20 0.36
TUBB2B Q9BVA1 1/20 0.36
TUBB1 Q9H4B7 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8645682 0.95 HSD17B3 (0.39) HSD17B3NOTUMALDH1A1MEN1KMT2A
SCHEMBL8644832 0.87 TUBB4A (0.37) HSD17B3ALDH1A1MEN1KMT2ATUBB4A
SCHEMBL8646116 0.85 GAA (0.42) ALDH1A1MEN1KMT2ATUBB4ATUBB
SCHEMBL8644828 0.84 TUBB4A (0.38) HSD17B3ALDH1A1MEN1KMT2ATUBB4A
SCHEMBL8646109 0.81 GAA (0.42) HSD17B3ALDH1A1MEN1KMT2ATUBB4A
SCHEMBL8645908 0.81 MAPT (0.35) NOTUMMAPTPOLBTP53
SCHEMBL8647255 0.81 TUBB4A (0.35) HSD17B3ALDH1A1KMT2ATUBB4ATUBB
SCHEMBL8645858 0.79 ALDH1A1 (0.42) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL8647250 0.78 TUBB4A (0.36) HSD17B3ALDH1A1KMT2ATUBB4ATUBB
SCHEMBL8645638 0.77 BRD4 (0.40) ALDH1A1MAPTPOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843972-A Heterocyclic β-adrenergic agonists PFIZER INC. (US) 1998-12-01 US disclosed
EP-0801060-A1 Heterocyclic Beta-3 Adrenergenic Agonists PFIZER INC. (US) 1997-10-15 EP disclosed