SCHEMBL8645908

SCHEMBL8645908

COC(=O)C1(C(=O)O)Cc2cc(CC(C)=O)ccc2N1C(C)=O

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.35
PTGS1 P23219 1/20 0.35
AKR1C3 P42330 1/20 0.35
AKR1C2 P52895 1/20 0.35
NOTUM Q6P988 1/20 0.34
TP53 P04637 1/20 0.33
FSHR P23945 1/20 0.33
LMNA P02545 9/20 0.32
POLB P06746 1/20 0.32
TACR1 P25103 1/20 0.32
TACR3 P29371 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8645900 0.95 MAPT (0.34) MAPTPTGS1AKR1C3AKR1C2NOTUM
SCHEMBL8648264 0.89 MAPT (0.33) MAPTPTGS1AKR1C3AKR1C2TP53
SCHEMBL8645861 0.88 MAPT (0.44) MAPTTP53LMNAPOLB
SCHEMBL8647457 0.86 LMNA (0.33) MAPTPTGS1AKR1C3AKR1C2NOTUM
SCHEMBL8647012 0.85 LMNA (0.33) MAPTPTGS1AKR1C3AKR1C2TP53
SCHEMBL8647266 0.84 KMT2A (0.37) LMNATACR1TACR3
SCHEMBL8645856 0.84 MAPT (0.40) MAPTTP53LMNAPOLB
SCHEMBL8647005 0.82 LMNA (0.34) MAPTNOTUMTP53LMNAPOLB
SCHEMBL8644950 0.82 AMPD2 (0.38) MAPTPOLBTACR1TACR3
SCHEMBL8645683 0.81 HSD17B3 (0.37) MAPTNOTUMTP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843972-A Heterocyclic β-adrenergic agonists PFIZER INC. (US) 1998-12-01 US disclosed
EP-0801060-A1 Heterocyclic Beta-3 Adrenergenic Agonists PFIZER INC. (US) 1997-10-15 EP disclosed