SCHEMBL8649474

SCHEMBL8649474

CS(C)=Nc1cccnc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.48
HTR3B O95264 1/20 0.48
HTR3A P46098 1/20 0.48
HTR3D Q70Z44 1/20 0.48
HTR3C Q8WXA8 1/20 0.48
NOS3 P29474 2/20 0.42
NOS1 P29475 2/20 0.42
NOS2 P35228 2/20 0.42
ALDH1A1 P00352 3/20 0.41
CYP2A6 P11509 3/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
MPI P34949 1/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HSP90AA1 P07900 1/20 0.37
MAPT P10636 4/20 0.36
KDM4E B2RXH2 3/20 0.36
LMNA P02545 2/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28755007 0.78 HTR3E (0.48) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL130894 0.75
SCHEMBL5174355 0.74 HTR3E (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL3284038 0.74 HTR3E (0.58) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL10905395 0.71 ALDH1A1 (0.45) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL9608571 0.70
SCHEMBL2477042 0.70
SCHEMBL2238457 0.70
SCHEMBL2477043 0.70
SCHEMBL3233290 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0598396-B1 Improved method for the preparation of 3-Amino-2-chloro-4-alkylpyridines BOEHRINGER INGELHEIM PHARMA (US) 1998-09-02 EP disclosed
US-5654429-A REACTING 3-AMINO-2-CHLOROPYRIDINE WITH A SULFIDE IN PRESENCE OF HALOGENATING AGENT, HEATING IN PRESENCE OF TRIETHYLAMINE, METHANESULFONIC ACID AND ORGANIC SOLVENT(OR PHENOL AND SOLVENT), THEN HEATING WITH ETHANOL AND RANEY NICKEL BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. 1997-08-05 US disclosed
EP-0598396-A1 Improved method for the preparation of 3-Amino-2-chloro-4-alkylpyridines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1994-05-25 EP disclosed