SCHEMBL8655419

SCHEMBL8655419

CC1=C(C(=O)O)C(C(C)C)C(C(=O)OCCN2CCN(Cc3cccnc3)CC2)=C(C)N1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 5/20 0.42
GAA P10253 2/20 0.42
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
CACNA1B Q00975 1/20 0.40
PKM P14618 1/20 0.40
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8797927 0.80 KMT2A (0.47) KDM4EALDH1A1GAAPKMMAPT
SCHEMBL8797726 0.78 CHRNA7 (0.48) KDM4EALDH1A1GAA
SCHEMBL8796974 0.77 CHRNA7 (0.45) KDM4EALDH1A1GAATDP1
SCHEMBL8655149 0.74 CHRNA7 (0.47) KDM4EALDH1A1GAATDP1CYP3A4
SCHEMBL8657345 0.72 CACNA1B (0.38) KDM4EALDH1A1CACNA1B
SCHEMBL8650566 0.71 ADORA3 (0.43) KDM4EALDH1A1GAACYP3A4CYP2C9
SCHEMBL8797115 0.71 CHRNA7 (0.50) KDM4EALDH1A1GAACYP3A4CYP2C9
SCHEMBL8796956 0.70 CHRNA7 (0.49) KDM4EALDH1A1GAACYP3A4CYP2C9
SCHEMBL10367116 0.70 CACNA1B (0.50) KDM4EALDH1A1GAATDP1CYP3A4
SCHEMBL8797447 0.69 CHRNA7 (0.46) KDM4EALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5843950-A 1,4-dihydropyridine compound and pharmaceutical composition containing the same NIKKEN CHEMICALS CO., LTD. (JP) 1998-12-01 US disclosed
EP-0801065-A1 1,4-DIHYDROPYRIDINE COMPOUND AND MEDICINAL COMPOSITION CONTAINING THE SAME Nikken Chemicals Company, Limited (JP) 1997-10-15 EP disclosed