SCHEMBL8661391

SCHEMBL8661391

CNS(=O)(=O)C(CC(N)=O)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP2C19 P33261 4/20 0.43
GABBR2 O75899 1/20 0.41
GABBR1 Q9UBS5 1/20 0.41
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
NPSR1 Q6W5P4 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
PKM P14618 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
SLC6A3 Q01959 3/20 0.39
DRD3 P35462 2/20 0.39
LMNA P02545 2/20 0.39
ADORA3 P0DMS8 1/20 0.39
EDNRB P24530 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658264 0.83 CYP2C19 (0.42) ALDH1A1CYP2C19GABBR2GABBR1PDE4A
SCHEMBL23174395 0.81 CYP2C19 (0.46) ALDH1A1CYP2C19GABBR2GABBR1PDE4A
SCHEMBL5998430 0.80 CYP2C19 (0.47) ALDH1A1CYP2C19GABBR2GABBR1NPSR1
SCHEMBL26136303 0.80 TAAR1 (0.44) ALDH1A1GABBR2GABBR1NPSR1SLC6A3
SCHEMBL28686570 0.77 TRPA1 (0.42) ALDH1A1CYP2C19PDE4APDE4BPDE4C
SCHEMBL19183147 0.75 SRC (0.47) ALDH1A1CYP2C19NPSR1CYP2D6SLC6A3
SCHEMBL5070388 0.75 SMN1; SMN2 (0.44) ALDH1A1CYP2C19NPSR1CYP1A2CYP2D6
SCHEMBL16348724 0.73 ALDH1A1 (0.56) ALDH1A1CYP2C19NPSR1CYP1A2CYP2D6
SCHEMBL16403447 0.71 NPSR1 (0.40) ALDH1A1NPSR1CYP1A2CYP2D6PKM
SCHEMBL5674838 0.71 ATM (0.49) ALDH1A1CYP2C19NPSR1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0625516-B1 Benzenesulphonamide derivatives for the treatment of bladder instability ZENECA LTD (GB) 1998-09-09 EP claimed
EP-0625516-A1 Benzenesulphonamide derivatives for the treatment of bladder instability ZENECA LIMITED (GB) 1994-11-23 EP claimed
EP-0625516-B1 Benzenesulphonamide derivatives for the treatment of bladder instability ZENECA LTD (GB) 1998-09-09 EP disclosed
EP-0625516-A1 Benzenesulphonamide derivatives for the treatment of bladder instability ZENECA LIMITED (GB) 1994-11-23 EP disclosed