SCHEMBL8661771

SCHEMBL8661771

[Li]c1cccc2c1C(CC#C)c1ccccc1-2

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.39
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
EPHX2 P34913 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8664361 0.80 HTR2A (0.52) HTR2ACA1CA2TSHR
SCHEMBL8587289 0.78 HTR2A (0.42) HTR2ACA1CA2EPHX2TSHR
SCHEMBL28613357 0.70 EDNRB (0.42) HTR2ACA1CA2TSHR
SCHEMBL7576966 0.65 HTR2A (0.64) HTR2ACA1CA2TSHR
SCHEMBL5569765 0.65 ACHE (0.33) HTR2A
SCHEMBL8719014 0.65 HTR2A (0.39) HTR2ACA1CA2
SCHEMBL9602938 0.65 GPR3 (0.34) HTR2A
SCHEMBL6544747 0.65 GPR3 (0.34) HTR2A
SCHEMBL7624908 0.63 HTR2A (0.45) HTR2ACA1CA2
SCHEMBL6545167 0.61 MEN1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5744666-A Process for preparing an alkynyl fulvene group containing compound and said compound PHILLIPS PETROLEUM COMPANY (US) 1998-04-28 US disclosed
US-5728908-A Process for preparing a bridged ligand and said bridged ligand PHILLIPS PETROLEUM COMPANY (US) 1998-03-17 US disclosed
US-5631203-A Metallocene compounds and preparation thereof containing terminal alkynes PHILLIPS PETROLEUM COMPANY (US) 1997-05-20 US disclosed