SCHEMBL8663086

SCHEMBL8663086

Cc1cc(NC(=O)NC(=O)c2c(F)cccc2F)c(C)c(Cl)c1Oc1ccc(C#N)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.43
KMT2A Q03164 4/20 0.43
KDM4E B2RXH2 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
MAPT P10636 2/20 0.37
USP2 O75604 1/20 0.37
ALOX15 P16050 1/20 0.37
MET P08581 3/20 0.37
ATM Q13315 1/20 0.35
AR P10275 3/20 0.34
GAA P10253 1/20 0.34
THRB P10828 1/20 0.34
RECQL P46063 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
BACE1 P56817 1/20 0.33
POLB P06746 1/20 0.33
GCK P35557 1/20 0.33
RORC P51449 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8658809 0.96 KDM4E (0.43) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL8659453 0.92 ALDH1A1 (0.36) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL8659385 0.91 TAS1R3 (0.40) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL8662513 0.87 MEN1 (0.45) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL8659984 0.86 KDR (0.42) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL8658919 0.85 PYGL (0.41) NPC1ARTDP1POLB
SCHEMBL8656628 0.85 MEN1 (0.45) MEN1KMT2AKDM4EMAPTUSP2
SCHEMBL8662606 0.85 S1PR3 (0.41) MEN1KMT2ANPC1ARPOLB
SCHEMBL9135451 0.84 MEN1 (0.41) MEN1KMT2AKDM4ENPC1ALDH1A1
SCHEMBL10639537 0.82 NPC1 (0.45) MEN1KMT2AKDM4ENPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5776981-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5776982-A Use of acyl urea compounds for controlling endoparasites and ectoparasites of warm-blooded animals NOVARTIS CORPORATION (US) 1998-07-07 US disclosed
US-5420163-A Insecticides or miticides CIBA-GEIGY (US) 1995-05-30 US disclosed
US-5135953-A Oral or injections; cattle, swine, poultry CIBA-GEIGY (US) 1992-08-04 US disclosed
EP-0115210-B1 PESTICIDAL BENZOYL UREAS AND PROCESS FOR THEIR PREPARATION UNION CARBIDE CORPORATION (US) 1988-05-11 EP disclosed
US-4659724-A Certain 1-[4-(5-cyano-2-pyridyloxy)phenyl-benzoyl ureas having pesticidal properties UNION CARBIDE CORPORATION (US) 1987-04-21 US disclosed
EP-0211004-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS RHONE-POULENC NEDERLAND B.V. (NL) 1987-02-25 EP disclosed
WO-1986003941-A1 USE OF ACYL UREA COMPOUNDS FOR CONTROLLING ENDOPARASITES AND ECTOPARASITES OF WARM-BLOODED ANIMALS UNION CARBIDE CORPORATION (US) 1986-07-17 WO disclosed
EP-0115210-A1 Pesticidal benzoyl ureas and process for their preparation UNION CARBIDE CORPORATION (US) 1984-08-08 EP disclosed