Oxyquinoline

Oxyquinoline

SCHEMBL866498

CC(N)=O.Oc1cccc2cccnc12

nearest known ligand 0.75

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.75
TSHR P16473 2/20 0.75
CHRM1 P11229 1/20 0.75
COMT P21964 1/20 0.75
ADRA1A P35348 1/20 0.75
METAP2 P50579 1/20 0.75
METAP1 P53582 1/20 0.75
HDAC8 Q9BY41 1/20 0.75
KDM4E B2RXH2 5/20 0.69
ALOX12 P18054 2/20 0.69
ALDH1A1 P00352 4/20 0.64
LMNA P02545 2/20 0.64
PARP1 P09874 1/20 0.59
PIM1 P11309 1/20 0.53
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
MAPK1 P28482 1/20 0.50
CA9 Q16790 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
TDP1 Q9NUW8 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxyquinoline SCHEMBL27477171 0.93 MMP2 (0.81) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL8605182 0.93 MMP2 (0.81) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL5965842 0.93 MMP2 (0.81) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL2867503 0.91 MMP2 (0.78) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL4465896 0.91 MMP2 (0.78) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL27553390 0.91 MMP2 (0.78) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL15568316 0.89 MMP2 (0.75) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL15568317 0.88 MMP2 (0.72) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL28459062 0.87 MMP2 (0.84) MMP2TSHRCHRM1COMTADRA1A
Oxyquinoline SCHEMBL28915558 0.87 TSHR (0.91) MMP2TSHRCHRM1COMTADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8058074-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-11-15 US claimed
US-20080044913-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF CHUNG-ANG UNIVERSITY INUDSTRY-ACADEMY COOPERATION FOUNDATION (KR) 2008-02-21 US claimed
US-20180017541-A1 SYSTEMS AND METHODS TO DETECT AND MEASURE MATERIALS IN OIL KINARD WILLIAM BRIAN (US) 2018-01-18 US disclosed
WO-2018013473-A1 SYSTEMS AND METHODS TO DETECT AND MEASURE MATERIALS IN OIL KINARD WILLIAM BRIAN (US) 2018-01-18 WO disclosed
US-8377698-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2013-02-19 US disclosed
US-8377698-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2013-02-19 US disclosed
US-8377698-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2013-02-19 US disclosed
US-20120077275-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF SAMSUNG ELECTRONICS CO.. LTD. (KR) 2012-03-29 US disclosed
US-20120077275-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF SAMSUNG ELECTRONICS CO.. LTD. (KR) 2012-03-29 US disclosed
US-8058074-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-11-15 US disclosed
US-8058074-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-11-15 US disclosed
US-8058074-B2 8-hydroxyquinoline acetamide compound, 8-hydroxy quinoline thioamide compound and use thereof SAMSUNG ELECTRONICS CO., LTD. (KR) 2011-11-15 US disclosed
US-20080044913-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF CHUNG-ANG UNIVERSITY INUDSTRY-ACADEMY COOPERATION FOUNDATION (KR) 2008-02-21 US disclosed
US-20080044913-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF CHUNG-ANG UNIVERSITY INUDSTRY-ACADEMY COOPERATION FOUNDATION (KR) 2008-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080044913-A1 NOVEL 8-HYDROXYQUINOLINE ACETAMIDE COMPOUND, 8-HYDROXY QUINOLINE THIOAMIDE COMPOUND AND USE THEREOF TST, TMT1A, HDHD5 MMP2 4479/4885TSHR 1983/4885CHRM1 2349/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.